| مستقبل الإستروجين | | الناهضات | 
- سترويدية: 2-Hydroxyestradiol
 
- 2-Hydroxyestrone
 
- 3-Methyl-19-methyleneandrosta-3,5-dien-17β-ol
 
- 3α-Androstanediol
 
- 3α,5α-Dihydrolevonorgestrel
 
- 3β,5α-Dihydrolevonorgestrel
 
- 3α-Hydroxytibolone
 
- 3β-Hydroxytibolone
 
- 3β-Androstanediol
 
- 4-Androstenediol
 
- 4-Androstenedione
 
- 4-Hydroxyestradiol
 
- 4-Hydroxyestrone
 
- 4-Methoxyestradiol
 
- 4-Methoxyestrone
 
- 5-Androstenediol
 
- 7-Oxo-DHEA
 
- 7α-Hydroxy-DHEA
 
- 7α-Methylestradiol
 
- 7β-Hydroxyepiandrosterone
 
- 8,9-Dehydroestradiol
 
- 8,9-Dehydroestrone
 
- 8β-VE2
 
- 10β,17β-Dihydroxyestra-1,4-dien-3-one (DHED)
 
- 16α-Fluoroestradiol
 
- 16α-Hydroxy-DHEA
 
- 16α-Hydroxyestrone
 
- 16α-Iodoestradiol
 
- 16α-LE2
 
- 16β,17α-Epiestriol (16β-hydroxy-17α-estradiol)
 
- 17α-Estradiol (alfatradiol)
 
- 17α-Dihydroequilenin
 
- 17α-Dihydroequilin
 
- 17α-Epiestriol (16α-hydroxy-17α-estradiol)
 
- 17β-Dihydroequilenin
 
- 17β-Dihydroequilin
 
- أبيراترون
 
- أسيستات الأبيراترون
 
- Alestramustine
 
- Almestrone
 
- ستروديات ابتنائية (مثل التستوستيرون والإسترات، methyltestosterone, metandienone (methandrostenolone), nandrolone and الإسترات، وغيرها كثير؛ via estrogenic metabolites)
 
- Atrimustine
 
- Bolandiol
 
- Bolandiol dipropionate
 
- Butolame
 
- Clomestrone
 
- Cloxestradiol
 
- Conjugated estrogens
 
- Cyclodiol
 
- Cyclotriol
 
- DHEA
 
- DHEA-S
 
- Epiestriol (16β-epiestriol, 16β-hydroxy-17β-estradiol)
 
- Epimestrol
 
- Equilenin
 
- Equilin
 
- ERA-63 (ORG-37663)
 
- Esterified estrogens
 
- Estetrol
 
- إستراديول
 
- Estramustine
 
- Estramustine phosphate
 
- Estrapronicate
 
- Estrazinol
 
- إستريول
 
- Estrofurate
 
- Estromustine
 
- إسترون
 
- Etamestrol (eptamestrol)
 
- Ethinylestradiol
 
- Ethinylestriol
 
- Ethylestradiol
 
- Etynodiol
 
- Etynodiol diacetate
 
- Hexolame
 
- Hippulin
 
- Hydroxyestrone diacetate
 
- Lynestrenol
 
- Lynestrenol phenylpropionate
 
- Mestranol
 
- Methylestradiol
 
- Moxestrol
 
- Mytatrienediol
 
- Nilestriol
 
- Norethisterone
 
- Noretynodrel
 
- Orestrate
 
- Pentolame
 
- Prodiame
 
- Prolame
 
- Promestriene
 
- RU-16117
 
- Quinestradol
 
- Quinestrol
 
- Tibolone
  
- Xenoestrogens: Anise-related (e.g., anethole, anol, dianethole, dianol, photoanethole)
 
- Chalconoids (e.g., isoliquiritigenin, phloretin, phlorizin (phloridzin), wedelolactone)
 
- Coumestans (e.g., coumestrol, psoralidin)
 
- Flavonoids (incl. 7,8-DHF, 8-prenylnaringenin, apigenin, baicalein, baicalin, biochanin A, calycosin, catechin, daidzein, daidzin, ECG, EGCG, epicatechin, equol, formononetin, glabrene, glabridin, genistein, genistin, glycitein, kaempferol, liquiritigenin, mirificin, myricetin, naringenin, penduletin, pinocembrin, prunetin, puerarin, quercetin, tectoridin, tectorigenin)
 
- Lavender oil
 
- Lignans (e.g., enterodiol, enterolactone, nyasol (cis-hinokiresinol))
 
- Metalloestrogens (مثل، كادميوم)
 
- Pesticides (e.g., alternariol, dieldrin, endosulfan, fenarimol, methiocarb, methoxychlor, triclocarban, triclosan)
 
- Phytosteroids (e.g., digitoxin (ديجيتالس), diosgenin, guggulsterone)
 
- الفايتوستيرولات (e.g., β-sitosterol, campesterol, stigmasterol)
 
- Resorcylic acid lactones (e.g., zearalanone, α-zearalenol, β-zearalenol, zearalenone, zeranol (α-zearalanol), taleranol (teranol, β-zearalanol))
 
- شبيهات السترويد (e.g., deoxymiroestrol, miroestrol)
 
- Stilbenoids (e.g., resveratrol, rhaponticin)
 
- Synthetic xenoestrogens (e.g., alkylphenols, bisphenols (e.g., BPA, BPF, BPS), DDT, parabens, PBBs, PHBA, فتالات، PCBs)
 
- Others (e.g., agnuside, rotundifuran)
  
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 منظمات مستقبل الإستروجية مختارة  مختلطة |  | 
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 | Antagonists | 
- Coregulator-binding modulators: ERX-11
  
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